Molecule Details
InChIKeyAOXRBFRFYPMWLR-XGXHKTLJSA-N
Compound NameEthylestrenol
Canonical SMILESCC[C@]1(O)CC[C@H]2[C@@H]3CCC4=CCCC[C@@H]4[C@H]3CC[C@@]21C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.83
SourceChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB01493
Drug NameEthylestrenol
CAS Number965-90-2
Groups approved withdrawn
ATC Codes A14AB02
DescriptionAn anabolic steroid with some progestational activity and little androgenic effect. [PubChem]

Categories: Alimentary Tract and Metabolism Anabolic Agents Anabolic Agents for Systemic Use Anabolic Steroids Estren Derivatives Fused-Ring Compounds Hormones Hormones, Hormone Substitutes, and Hormone Antagonists Norpregnanes Norpregnenes Norsteroids Steroids
Cross-references: ChEBI: 31578 CHEMBL1200623 ChemSpider: 13168 PharmGKB: PA449539 PubChem:13765 PubChem:46505460 RxCUI: 4162 Wikipedia: Ethylestrenol ZINC: ZINC000004215863
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.2 IC50 ChEMBL
P08172 CHRM2 Homo sapiens Human PF00001 6.8 IC50 ChEMBL
P03372 ESR1 Homo sapiens Human PF12743 PF00104 PF02159 PF00105 6.5 Ki ChEMBL
DrugBank Target Actions (1)
Target Gene Target Name Action Type
P10275 AR Androgen receptor modulator targets