Molecule Details
InChIKeyAOLQSKKQHIKRMB-UHFFFAOYSA-N
Compound Namen-[3-(5-Amino-1-pyridin-2-yl-1h-[1,2,4]triazol-3-ylamino)-phenyl]-acetamide
Canonical SMILESCC(=O)Nc1cccc(Nc2nc(N)n(-c3ccccn3)n2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.61
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 8.1 Ki ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 8.1 pIC50 TTD_MultiTarget
P10721 KIT Homo sapiens Human PF00047 PF07714 6.7 Ki ChEMBL;BindingDB