Target not found.
Molecule Details
InChIKeyAOGOUTMDEVCZHA-UHFFFAOYSA-N
Compound Name2-{4-[(4-Hydroxy-quinazolin-6-ylmethyl)-prop-2-ynyl-amino]-benzoylamino}-pentanedioic acid
Canonical SMILESC#CCN(Cc1ccc2ncnc(O)c2c1)c1ccc(C(=O)NC(CCC(=O)O)C(=O)O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.32
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 7.6 pIC50 TTD_MultiTarget
P04818 TYMS Homo sapiens Human PF00303 7.6 Ki ChEMBL;BindingDB
P00469 thyA Lacticaseibacillus casei Pathogen PF00303 6.8 IC50 ChEMBL;BindingDB