Molecule Details
InChIKeyANZIISNSHPKVRV-UHFFFAOYSA-N
Compound NameAbanoquil
Canonical SMILESCOc1cc2c(cc1OC)CN(c1cc(N)c3cc(OC)c(OC)cc3n1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL10.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB20666
Drug NameAbanoquil
CAS Number90402-40-7
Groups experimental
ATC Codes nan
DescriptionAbanoquil is a small molecule drug. Abanoquil has a monoisotopic molecular weight of 395.18 Da.

Categories: Heterocyclic Compounds, Fused-Ring Isoquinolines Quinolines
Cross-references: BindingDB: 50033109 CHEMBL324090
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25100 ADRA1D Homo sapiens Human PF00001 10.4 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 10.4 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 10.0 Ki ChEMBL;BindingDB
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P25100 ADRA1D Alpha-1D adrenergic receptor inhibitor targets
P35348 ADRA1A Alpha-1A adrenergic receptor inhibitor targets
P35368 ADRA1B Alpha-1B adrenergic receptor inhibitor targets