Molecule Details
InChIKeyANDYPXVQXOKMKT-UHFFFAOYSA-N
Compound Name5-fluoro-4-(8-fluoro-4-propan-2-yl-2,3-dihydro-1,4-benzoxazin-6-yl)-N-[5-(3-methylpiperazin-1-yl)-2-pyridinyl]pyrimidin-2-amine
Canonical SMILESCC1CN(c2ccc(Nc3ncc(F)c(-c4cc(F)c5c(c4)N(C(C)C)CCO5)n3)nc2)CCN1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00534 CDK6 Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 6.2 IC50 ChEMBL;BindingDB