Molecule Details
InChIKeyANAOYTVZYSRWRF-HNNXBMFYSA-N
Compound Name6-[6-(6-methylpyrazin-2-yl)pyrazolo[4,3-c]pyridin-1-yl]-2-[(3S)-piperidin-3-yl]pyridazin-3-one
Canonical SMILESCc1cncc(-c2cc3c(cn2)cnn3-c2ccc(=O)n([C@H]3CCCNC3)n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.9 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.6 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.7 Ki ChEMBL;BindingDB