Molecule Details
InChIKeyANAMVZJDWRVIRM-KEEVHDRGSA-N
Compound Name(10R,14S)-14-[4-[5-chloro-2-(3-methyl-1,2,4-triazol-1-yl)phenyl]-6-oxo-2,3-dihydropyridin-1-yl]-10-methyl-8,16-diazatricyclo[13.3.1.02,7]nonadeca-1(19),2,4,6,15,17-hexaen-9-one
Canonical SMILESCc1ncn(-c2ccc(Cl)cc2C2=CC(=O)N([C@H]3CCC[C@@H](C)C(=O)Nc4ccccc4-c4ccnc3c4)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00740 F9 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.4 Ki ChEMBL;BindingDB
P03951 F11 Homo sapiens Human PF00024 PF00089 7.4 Ki ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 6.6 Ki ChEMBL;BindingDB