Molecule Details
InChIKeyALZQLPXUMAEFBO-HOTGVXAUSA-N
Compound Name(R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-mercapto-2-(3-phenyl-ureido)-propionamide
Canonical SMILESNC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CS)NC(=O)Nc1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.59
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.0 IC50 ChEMBL;BindingDB
P03956 MMP1 Homo sapiens Human PF00045 PF00413 PF01471 7.4 IC50 ChEMBL;BindingDB
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 7.4 pIC50 TTD_MultiTarget