Molecule Details
InChIKeyALJJNAMKZDVVQD-UHFFFAOYSA-N
Compound Name[2-(7-Fluoro-2,3-dihydro-benzo[1,4]dioxin-5-yloxy)-ethyl]-[3-(5-fluoro-1H-indol-3-yl)-propyl]-amine
Canonical SMILESFc1cc(OCCNCCCc2c[nH]c3ccc(F)cc23)c2c(c1)OCCO2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.21
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.6 IC50 ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 Clinical TTD_MultiTarget TTD_MultiTarget