Molecule Details
InChIKeyALGIYGCMWHXAJQ-UHFFFAOYSA-N
Compound Name4-[(1,3-dimethylpyrazolo[4,5-e][1,2,4]triazin-5-yl)amino]-N-(2-morpholin-4-ylethyl)benzenesulfonamide
Canonical SMILESCc1nn(C)c2nnc(Nc3ccc(S(=O)(=O)NCCN4CCOCC4)cc3)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 8.2 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB