Molecule Details
InChIKeyAKUJIVTZSHCXRK-HNNXBMFYSA-N
Compound NameUS10155760, Example 10
Canonical SMILESCC(=O)Nc1cc(-c2cc(F)c(OC[C@@H](N)CC(C)C)c(Cl)c2)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q2M2I8 AAK1 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.1 IC50 ChEMBL