Molecule Details
InChIKeyAKTXUNFJKSXMRB-UHFFFAOYSA-N
Compound Name7-(4-Fluorophenyl)-2-(2-methoxyethyl)-8-(3-met hylimidazo[1,2-a]pyridin-6-yl)-[1,2,4]triazolo[1, 5-c]pyrimidin-5-amine
Canonical SMILESCOCCc1nc2c(-c3ccc4ncc(C)n4c3)c(-c3ccc(F)cc3)nc(N)n2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.44
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.7 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB