Molecule Details
InChIKeyAJLZQJOCQFFRQL-UHFFFAOYSA-N
Compound NameN-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-4-[(2-methyl-6-propan-2-ylthieno[2,3-d]pyrimidin-4-yl)amino]-1H-pyrazole-5-carboxamide
Canonical SMILESCc1nc(Nc2c[nH]nc2C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c2cc(C(C)C)sc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 9.1 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB