Molecule Details
InChIKeyAIGFEVGWAQPOEK-MOPGFXCFSA-N
Compound Name(3R,5S)-1-benzyl-6-methoxy-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Canonical SMILESCOc1cccc2c1[C@H](C)N(C(=O)Nc1cccnc1)[C@H](C)CN2Cc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P0X4 CACNA1I Homo sapiens Human PF00520 6.9 IC50 ChEMBL;BindingDB
O43497 CACNA1G Homo sapiens Human PF00520 6.7 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 6.5 IC50 ChEMBL;BindingDB