Molecule Details
InChIKeyAIDWTYRIDDCANO-UHFFFAOYSA-N
Compound Name3-[5-(Piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-1,2,3-triazol-1-yl)-1h-indazole
Canonical SMILESc1cn(-c2ccc3c(-c4cc5cc(CN6CCCCC6)ccc5[nH]4)n[nH]c3c2)nn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.69
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14757 CHEK1 Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P50613 CDK7 Homo sapiens Human PF00069 7.2 IC50 ChEMBL
P51946 CCNH Homo sapiens Human PF16899 PF00134 7.2 IC50 BindingDB