Molecule Details
InChIKeyAHYGIWNTGDKMRR-SUAIOLNFSA-N
Compound Name(2S)-2-[(3S)-4-[(2R)-3-(4-fluorophenyl)-2-[[(2S)-2-(methylamino)propanoyl]amino]propanoyl]-2-oxo-3-propylpiperazin-1-yl]-N-methyl-3-naphthalen-2-ylpropanamide
Canonical SMILESCCC[C@H]1C(=O)N([C@@H](Cc2ccc3ccccc3c2)C(=O)NC)CCN1C(=O)[C@@H](Cc1ccc(F)cc1)NC(=O)[C@H](C)NC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
Q01726 MC1R Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB