Molecule Details
InChIKeyAHFARWUGWOGTLO-UHFFFAOYSA-N
Compound NameN,N-dimethyl-2-[4-[4-(2-methyl-3-propan-2-ylbenzimidazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide
Canonical SMILESCc1nc2ccc(-c3ccnc4[nH]c(C5CCN(CC(=O)N(C)C)CC5)cc34)cc2n1C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50750 CDK9 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB