Molecule Details
InChIKeyAHEMFHZQUVEVBH-UHFFFAOYSA-N
Compound Name3,4-Dichloro-2-iodo-1-(1-methylpiperidin-4-yl)pyrrolo[2,3-b]pyridine-6-carboxamide
Canonical SMILESCN1CCC(n2c(I)c(Cl)c3c(Cl)cc(C(N)=O)nc32)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB