Molecule Details
InChIKeyAGNYFINNIVFBHA-UHFFFAOYSA-N
Compound Name1-(3-{[2,6-Dimethyl-5-methylcarbamoyl-4-(4-nitro-phenyl)-1,4-dihydro-pyridine-3-carbonyl]-amino}-propyl)-4-phenyl-piperidine-4-carboxylic acid methyl ester
Canonical SMILESCNC(=O)C1C(C)=NC(C)=C(C(=O)NCCCN2CCC(C(=O)OC)(c3ccccc3)CC2)C1c1ccc([N+](=O)[O-])cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL6.8
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 8.4 Ki BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.4 Ki BindingDB
P35367 HRH1 Homo sapiens Human PF00001 6.3 Ki BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 6.1 Ki BindingDB