Molecule Details
InChIKeyAFUSGLDYQSDIEU-NQIIRXRSSA-N
Compound Name(2s,4r)-1-(3-Amino-2-Methylbenzoyl)-4-Hydroxy-N-(4-(4-Methylthiazol-5-Yl)benzyl)pyrrolidine-2-Carboxamide
Canonical SMILESCc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)c2cccc(N)c2C)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P40337 VHL Homo sapiens Human PF01847 PF17211 6.0 IC50 ChEMBL;BindingDB
Q15369 ELOC Homo sapiens Human PF03931 6.0 IC50 ChEMBL;BindingDB
Q15370 ELOB Homo sapiens Human PF00240 6.0 IC50 ChEMBL