Molecule Details
InChIKeyADXFJIYJEFFOSY-UHFFFAOYSA-N
Compound Name1-(1-{3-[1-Benzyl-3-(3,4-dichloro-phenyl)-6-oxo-piperidin-3-yl]-propyl}-piperidin-4-yl)-1,3-dihydro-benzoimidazol-2-one
Canonical SMILESO=C1CCC(CCCN2CCC(n3c(=O)[nH]c4ccccc43)CC2)(c2ccc(Cl)c(Cl)c2)CN1Cc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21452 TACR2 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P29371 TACR3 Homo sapiens Human PF00001 6.3 IC50 ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB