Molecule Details
InChIKeyADBUMAAMWCLEEI-UHFFFAOYSA-N
Compound Name2-(1H-Benzoimidazol-5-yl)-N-(5-cyclobutyl-thiazol-2-yl)-acetamide
Canonical SMILESO=C(Cc1ccc2[nH]cnc2c1)Nc1ncc(C2CCC2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00535 CDK5 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 7.5 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB