Molecule Details
InChIKeyACXZKUHGYNILFP-UHFFFAOYSA-N
Compound Name2-[[4-[(2,4-Diaminofuro[2,3-d]pyrimidin-5-yl)methylamino]benzoyl]amino]pentanedioic acid
Canonical SMILESNc1nc(N)c2c(CNc3ccc(C(=O)NC(CCC(=O)O)C(=O)O)cc3)coc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.3 IC50 ChEMBL;BindingDB
P00381 folA Lacticaseibacillus casei Pathogen PF00186 6.2 IC50 ChEMBL;BindingDB
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 6.2 IC50 ChEMBL;BindingDB