Molecule Details
InChIKeyACILVPXHSUHXNS-UHFFFAOYSA-N
Compound Name1-[5-[3-([1,2,4]Triazolo[1,5-a]pyrimidin-7-yl)piperidine-1-carbonyl]indol-1-yl]ethanone
Canonical SMILESCC(=O)n1ccc2cc(C(=O)N3CCCC(c4ccnc5ncnn45)C3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O00408 PDE2A Homo sapiens Human PF01590 PF00233 8.7 IC50 ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 6.5 IC50 ChEMBL;BindingDB