Molecule Details
InChIKeyACHQQXOLWIKHRK-UHFFFAOYSA-N
Compound Name2-[4-(3,4-Dichlorophenyl)piperazin-1-ylmethyl]-6-(piperidin-1-yl)imidazo[1,2-b]pyridazine
Canonical SMILESClc1ccc(N2CCN(Cc3cn4nc(N5CCCCC5)ccc4n3)CC2)cc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB