Molecule Details
InChIKeyACGBFWCBVIXTPZ-NBEIKUQISA-N
Canonical SMILESCO[C@H]1CC[C@@H](C(=O)Nc2cc(-c3ccnc(Nc4ccc(F)cc4)c3)ccn2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB