Molecule Details
InChIKeyACDQVXJNZDLXFP-UHFFFAOYSA-N
Compound NameN-(4-cyano-3-(thiazol-2-yl)thiophen-2-yl)-2-(2-oxo-6-(trifluoromethyl)quinolin-1(2H)-yl)acetamide
Canonical SMILESN#Cc1csc(NC(=O)Cn2c(=O)ccc3cc(C(F)(F)F)ccc32)c1-c1nccs1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.83
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB