Molecule Details
InChIKeyABNXKGFLZFSILK-MOPGFXCFSA-N
Canonical SMILESO=C(O)C[C@H](NC(=O)[C@@H]1CCCN(C(=O)CCC2CCNCC2)C1)c1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB21212
Drug NameElarofiban anhydrous
CAS Number198958-88-2
Groups experimental
ATC Codes nan
DescriptionElarofiban anhydrous is a small molecule drug. The usage of the INN stem '-fiban' in the name indicates that Elarofiban anhydrous is a fibrinogen receptor antagonist (glycoprotein IIb/IIIa receptor antagonist). Elarofiban anhydrous has a monoisotopic molecular weight of 416.24 Da.

Categories: Piperidines
Cross-references: BindingDB: 50104600 CHEMBL87728
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P05106 ITGB3 Homo sapiens Human PF07974 PF23105 PF18372 PF08725 PF07965 PF00362 PF17205 9.8 IC50 ChEMBL
P08514 ITGA2B Homo sapiens Human PF01839 PF08441 PF20805 PF20806 PF00357 9.8 IC50 ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P05106 ITGB3 Integrin beta-3 modulator targets
P08514 ITGA2B Integrin alpha-IIb modulator targets