Molecule Details
InChIKeyABJKWBDEJIDSJZ-UHFFFAOYSA-N
Canonical SMILESCN(Cc1ccc(C(C)(C)C)cc1)Cc1cccc2ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.32
SourceChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB01091
Drug NameButenafine
CAS Number101828-21-1
Groups approved
ATC Codes D01AE23
DescriptionButenafine hydrochloride is a synthetic benzylamine antifungal agent. Butenafine's mechanism of action is believed to involve the synthesis inhibition of sterols. In particular, butenafine acts to inhibit the activity of the squalene epoxidase enzyme that is essential in the formation of sterols nec...

Categories: Amines Anti-Infective Agents Antifungal Agents Antifungals for Dermatological Use Antifungals for Topical Use Benzene Derivatives Benzyl Compounds Benzylamine Antifungal Benzylamines Dermatologicals
Cross-references: BindingDB: 50436713 ChEBI: 3238 CHEMBL990 ChemSpider: 2390 Drugs Product Database (DPD): 11423 C08067 D07596 PharmGKB: PA164745478 PubChem:2484 PubChem:46506191 RxCUI: 47461 Therapeutic Targets Database: DAP001236 Wikipedia: Butenafine ZINC: ZINC000001530975
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10635 CYP2D6 Homo sapiens Human PF00067 6.5 IC50 ChEMBL
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 6.1 Ki ChEMBL
DrugBank Target Actions (2)
Target Gene Target Name Action Type
Q14534 SQLE Squalene monooxygenase inhibitor targets
Q92206 ERG1 Squalene epoxidase ERG1 modulator targets