Molecule Details
InChIKeyABFNTRQPWNXUHA-UBKPHHHOSA-N
Compound Name2-[(3R,6S,9R,12R,15R,18S)-9-(4-aminobutyl)-3,18-dibenzyl-6-[(1R)-1-hydroxyethyl]-12,15-bis(1H-indol-3-ylmethyl)-2,5,8,11,14,17,20,25-octaoxo-1,4,7,10,13,16,19,24-octazacyclooctacos-1-yl]acetamide
Canonical SMILESC[C@@H](O)[C@@H]1NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)CCCNC(=O)CCCN(CC(N)=O)C(=O)[C@@H](Cc2ccccc2)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35346 SSTR5 Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P30874 SSTR2 Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB
P31391 SSTR4 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB