Molecule Details
InChIKeyABAZYTXCHHQMTO-UHFFFAOYSA-N
Compound NameN-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-6-[3-(methylamino)phenyl]-2-oxo-3-[(2-phenylethyl)amino]-1,2-dihydropyrazin-1-yl}acetamide
Canonical SMILESCNc1cccc(-c2c(Cl)nc(NCCc3ccccc3)c(=O)n2CC(=O)NCc2ccc(C(=N)N)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.2 IC50 ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.2 IC50 ChEMBL;BindingDB
P13726 F3 Homo sapiens Human PF09294 PF01108 6.2 IC50 ChEMBL