Molecule Details
InChIKeyAAYWXOINDKYXKL-UHFFFAOYSA-N
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCN(CC[N+](C)(C)[O-])C5)ncc3F)cc2n1C1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB