Molecule Details
InChIKeyAAXGNXOJOSOUQQ-SANMLTNESA-N
Compound Name4-(5-{[(1-Benzyl-2-oxo-pyrrolidin-3-yl)-butyl-amino]-methyl}-imidazol-1-ylmethyl)-benzonitrile
Canonical SMILESCCCCN(Cc1cncn1Cc1ccc(C#N)cc1)[C@H]1CCN(Cc2ccccc2)C1=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.14
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.4 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.3 IC50 ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.7 IC50 ChEMBL;BindingDB