Molecule Details
InChIKeyAAMUKYFUFDUBDC-JTQLQIEISA-N
Compound Name2-N-[(1S)-1-(3-chloro-1H-pyrrolo[3,2-b]pyridin-5-yl)ethyl]-4-N-(5-cyclopropyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine
Canonical SMILESC[C@H](Nc1nccc(Nc2cc(C3CC3)[nH]n2)n1)c1ccc2[nH]cc(Cl)c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13153 PAK1 Homo sapiens Human PF00786 PF00069 8.2 Ki ChEMBL;BindingDB
O75914 PAK3 Homo sapiens Human PF00786 PF00069 6.8 IC50 ChEMBL
Q13177 PAK2 Homo sapiens Human PF00786 PF00069 6.8 IC50 ChEMBL