Molecule Details
InChIKeyAAADQEFQWNJHOZ-UHFFFAOYSA-N
Compound Name5-(4-Chloro-phenyl)-9-fluoro-2,5-dihydro-3H-imidazo[2,1-a]isoindol-5-ol
Canonical SMILESOC1(c2ccc(Cl)cc2)c2cccc(F)c2C2=NCCN21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P23975 SLC6A2 Homo sapiens Human PF00209 8.7 IC50 ChEMBL;BindingDB
Q01959 SLC6A3 Homo sapiens Human PF00209 7.6 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.2 IC50 ChEMBL;BindingDB