Transcriptional misregulation in cancer

hsa05202 79 targets in this pathway

UniProt AC Gene Protein Name Organism Multi-Target Molecules
Q13547 HDAC1 Histone deacetylase 1 Homo sapiens 5940 Detail
Q92769 HDAC2 Histone deacetylase 2 Homo sapiens 3821 Detail
P50750 CDK9 Cyclin-dependent kinase 9 Homo sapiens 3102 Detail
O60563 CCNT1 Cyclin-T1 Homo sapiens 2851 Detail
P36888 FLT3 Receptor-type tyrosine-protein kinase FLT3 Homo sapiens 2188 Detail
P14780 MMP9 Matrix metalloproteinase-9 Homo sapiens 1941 Detail
P20248 CCNA2 Cyclin-A2 Homo sapiens 1415 Detail
Q00987 MDM2 E3 ubiquitin-protein ligase Mdm2 Homo sapiens 1334 Detail
P08254 MMP3 Stromelysin-1 Homo sapiens 1292 Detail
P17948 FLT1 Vascular endothelial growth factor receptor 1 Homo sapiens 1237 Detail
P04637 TP53 Cellular tumor antigen p53 Homo sapiens 1173 Detail
P04629 NTRK1 High affinity nerve growth factor receptor Homo sapiens 1127 Detail
P08581 MET Hepatocyte growth factor receptor Homo sapiens 1125 Detail
Q07817 BCL2L1 Bcl-2-like protein 1 Homo sapiens 990 Detail
P07333 CSF1R Macrophage colony-stimulating factor 1 receptor Homo sapiens 896 Detail
Q13490 BIRC2 Baculoviral IAP repeat-containing protein 2 Homo sapiens 876 Detail
P78396 CCNA1 Cyclin-A1 Homo sapiens 730 Detail
P19793 RXRA Retinoic acid receptor RXR-alpha Homo sapiens 702 Detail
P08069 IGF1R Insulin-like growth factor 1 receptor Homo sapiens 611 Detail
Q13489 BIRC3 Baculoviral IAP repeat-containing protein 3 Homo sapiens 532 Detail
P41182 BCL6 B-cell lymphoma 6 protein Homo sapiens 472 Detail
P37231 PPARG Peroxisome proliferator-activated receptor gamma Homo sapiens 417 Detail
P26010 ITGB7 Integrin beta-7 Homo sapiens 355 Detail
Q05397 PTK2 Focal adhesion kinase 1 Homo sapiens 325 Detail
P00749 PLAU Urokinase-type plasminogen activator Homo sapiens 256 Detail
Q03164 KMT2A Histone-lysine N-methyltransferase 2A Homo sapiens 252 Detail
Q13315 ATM Serine-protein kinase ATM Homo sapiens 170 Detail
O00255 MEN1 Menin Homo sapiens 147 Detail
P37173 TGFBR2 TGF-beta receptor type-2 Homo sapiens 144 Detail
P19838 NFKB1 Nuclear factor NF-kappa-B p105 subunit Homo sapiens 140 Detail
Q04206 RELA Transcription factor p65 Homo sapiens 134 Detail
Q9NSY1 BMP2K BMP-2-inducible protein kinase Homo sapiens 111 Detail
P10276 RARA Retinoic acid receptor alpha Homo sapiens 108 Detail
P00750 PLAT Tissue-type plasminogen activator Homo sapiens 95 Detail
P48443 RXRG Retinoic acid receptor RXR-gamma Homo sapiens 94 Detail
P42263 GRIA3 Glutamate receptor 3 Homo sapiens 93 Detail
P08246 ELANE Neutrophil elastase Homo sapiens 90 Detail
O94921 CDK14 Cyclin-dependent kinase 14 Homo sapiens 90 Detail
P05164 MPO Myeloperoxidase Homo sapiens 87 Detail
P28702 RXRB Retinoic acid receptor RXR-beta Homo sapiens 87 Detail
P30279 CCND2 G1/S-specific cyclin-D2 Homo sapiens 71 Detail
Q16548 BCL2A1 Bcl-2-related protein A1 Homo sapiens 59 Detail
O75376 NCOR1 Nuclear receptor corepressor 1 Homo sapiens 58 Detail
P15428 HPGD 15-hydroxyprostaglandin dehydrogenase [NAD(+)] Homo sapiens 39 Detail
Q15532 SS18 Protein SSXT Homo sapiens 38 Detail
O15393 TMPRSS2 Transmembrane protease serine 2 Homo sapiens 37 Detail
Q03111 MLLT1 Protein ENL Homo sapiens 34 Detail
P42568 MLLT3 Protein AF-9 Homo sapiens 32 Detail
O96028 NSD2 Histone-lysine N-methyltransferase NSD2 Homo sapiens 29 Detail
P41212 ETV6 Transcription factor ETV6 Homo sapiens 19 Detail
P01106 MYC Myc proto-oncogene protein Homo sapiens 19 Detail
P05231 IL6 Interleukin-6 Homo sapiens 17 Detail
Q01196 RUNX1 Runt-related transcription factor 1 Homo sapiens 11 Detail
P10145 CXCL8 Interleukin-8 Homo sapiens 9 Detail
O60583 CCNT2 Cyclin-T2 Homo sapiens 9 Detail
P18846 ATF1 Cyclic AMP-dependent transcription factor ATF-1 Homo sapiens 8 Detail
Q8TEK3 DOT1L Histone-lysine N-methyltransferase, H3 lysine-79 specific Homo sapiens 7 Detail
Q16611 BAK1 Bcl-2 homologous antagonist/killer Homo sapiens 6 Detail
Q01844 EWSR1 RNA-binding protein EWS Homo sapiens 5 Detail
Q01543 FLI1 Friend leukemia integration 1 transcription factor Homo sapiens 5 Detail
P04141 CSF2 Granulocyte-macrophage colony-stimulating factor Homo sapiens 4 Detail
P10144 GZMB Granzyme B Homo sapiens 4 Detail
Q92570 NR4A3 Nuclear receptor subfamily 4 group A member 3 Homo sapiens 4 Detail
P25942 CD40 Tumor necrosis factor receptor superfamily member 5 Homo sapiens 4 Detail
P17844 DDX5 Probable ATP-dependent RNA helicase DDX5 Homo sapiens 3 Detail
P68431 H3C1 Histone H3.1 Homo sapiens 3 Detail
P35637 FUS RNA-binding protein FUS Homo sapiens 2 Detail
P11215 ITGAM Integrin alpha-M Homo sapiens 2 Detail
O15550 KDM6A Lysine-specific demethylase 6A Homo sapiens 2 Detail
P08571 CD14 Monocyte differentiation antigen CD14 Homo sapiens 2 Detail
P38936 CDKN1A Cyclin-dependent kinase inhibitor 1 Homo sapiens 1 Detail
Q16828 DUSP6 Dual specificity protein phosphatase 6 Homo sapiens 1 Detail
P11308 ERG Transcriptional regulator ERG Homo sapiens 1 Detail
Q96ST3 SIN3A Paired amphipathic helix protein Sin3a Homo sapiens 1 Detail
P61244 MAX Protein max Homo sapiens 1 Detail
P51825 AFF1 AF4/FMR2 family member 1 Homo sapiens 1 Detail
P04085 PDGFA Platelet-derived growth factor subunit A Homo sapiens 1 Detail
Q07812 BAX Apoptosis regulator BAX Homo sapiens 1 Detail
Q92804 TAF15 TATA-binding protein-associated factor 2N Homo sapiens 1 Detail